FILES containd dataset for paper: Characterization of new, efficient Mycobacterium tuberculosis topoisomerase-I inhibitors and their interaction with human ABC multidrug transporters Csilla Temesszentandrási-Ambrus1,2, Balázs Sarkadi1, Gergely Szakács1, Szilárd Tóth1, László Őrfi3,4, Csaba Szántai-Kis3, Péter Bánhegyi3, István Szabadkai3, Ferenc Baska3, Ruben C. Hartkoorn5, Rinkee Verma6, Valakunja Nagaraja6, Mary A Lingerfelt 7, Sean Ekins7 and Ágnes Telbisz1,* This work is dedicated to late Prof. György Kéri, founder and CEO of Vichem Ltd. 1 Institute of Enzymology, RCNS-HAS, Budapest, Hungary 2 Molecular Medicine Doctoral School, Semmelweis University, Budapest, Hungary 3 Vichem Chemie Research Ltd., Budapest, Hungary. 4 Department of Pharmaceutical Chemistry, Semmelweis University, Budapest, Hungary 5 Chemical Biology of Antibiotics, Center for Infection and Immunity, Inserm, CNRS, Institut Pasteur de Lille, Université de Lille, Lille, France 6 Department of Microbiology and Cell Biology, Indian Institute of Science, Bangalore, India 7 Collaborations Pharmaceuticals, Inc., 840 Main Campus Drive, Lab 3510, Raleigh, USA *Corresponding author: e-mail: telbisz.agnes@ttk.mta.hu