Estrogen receptor ligands. Part 9: Dihydrobenzoxathiin SERAMs with alkyl substituted pyrrolidine side chains and linkers
Copyright policy ) Timothy A, Blizzard; Frank, Dininno; Jerry D, Morgan; Helen Y, Chen; Jane Y, Wu; Seongkon, Kim; Wanda, Chan; +13 Authors
Timothy A, Blizzard; Frank, Dininno; Jerry D, Morgan; Helen Y, Chen; Jane Y, Wu; Seongkon, Kim; Wanda, Chan; Elizabeth T, Birzin; Yi Tien, Yang; Lee-Yuh, Pai; Paula M D, Fitzgerald; Nandini, Sharma; Ying, Li; Zhoupeng, Zhang; Edward C, Hayes; Carolyn A, Dasilva; Wei, Tang; Susan P, Rohrer; James M, Schaeffer; Milton L, Hammond;
Estrogen receptor ligands. Part 9: Dihydrobenzoxathiin SERAMs with alkyl substituted pyrrolidine side chains and linkers
A series of dihydrobenzoxathiin SERAMs with alkylated pyrrolidine side chains or alkylated linkers was prepared. Minor modifications in the side chain or linker resulted in significant effects on biological activity, especially in uterine tissue.
- Merck & Co. United States
Models, Molecular, Oxathiins, Selective Estrogen Receptor Modulators, Pyrrolidines, Receptors, Estrogen, Ligands
Models, Molecular, Oxathiins, Selective Estrogen Receptor Modulators, Pyrrolidines, Receptors, Estrogen, Ligands
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selected citations
Citations provided by BIP!
These citations are derived from selected sources.
This is an alternative to the "Influence" indicator, which also reflects the overall/total impact of an article in the research community at large, based on the underlying citation network (diachronically).
Citations provided by BIP!popularityPopularity provided by BIP!
This indicator reflects the "current" impact/attention (the "hype") of an article in the research community at large, based on the underlying citation network.
Popularity provided by BIP! 62
Top 10%
Top 10%
Top 10%
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