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image/svg+xml Jakob Voss, based on art designer at PLoS, modified by Wikipedia users Nina and Beao Closed Access logo, derived from PLoS Open Access logo. This version with transparent background. http://commons.wikimedia.org/wiki/File:Closed_Access_logo_transparent.svg Jakob Voss, based on art designer at PLoS, modified by Wikipedia users Nina and Beao Bioorganic & Medicin...arrow_drop_down
image/svg+xml Jakob Voss, based on art designer at PLoS, modified by Wikipedia users Nina and Beao Closed Access logo, derived from PLoS Open Access logo. This version with transparent background. http://commons.wikimedia.org/wiki/File:Closed_Access_logo_transparent.svg Jakob Voss, based on art designer at PLoS, modified by Wikipedia users Nina and Beao
Bioorganic & Medicinal Chemistry Letters
Article . 2012 . Peer-reviewed
License: Elsevier TDM
Data sources: Crossref
https://pubmed.ncbi.nlm.nih.go...
Article . 2013
Data sources: Europe PubMed Central
https://dx.doi.org/10.1016/j.b...
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Formylated polyamines as peptidomimetics

descriptionPublicationkeyboard_double_arrow_right Article 01 Nov 2012 English Publisher:Elsevier BVJournal:Bioorganic & Medicinal Chemistry Letters, volume 22, pages 6,580-6,582 (issn: 0960-894X, Copyright policy )
Authors: Sacha, Javor; Aaron, Janowsky; Robert, Johnson; Katherine, Wolfrum; Mitra, Tadayoni-Rebek; Julius, Rebek;

doi: 10.1016/j.bmcl.2012.09.008

pmid: 23017884

Formylated polyamines as peptidomimetics

Abstract

A new construct for imitating a natural peptide ligand using a modified retro-inverso sequence is described. It is demonstrated through the synthesis of a peptidomimetic derived from the endogenous sequence of leucine enkephalin. The product was active at 400 nM and selective for μ-opioid receptors.

Related Organizations
Keywords

Molecular Structure, Polyamines, Receptors, Opioid, mu, Biological Availability, Humans, Peptidomimetics

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selected citations
These citations are derived from selected sources.
This is an alternative to the "Influence" indicator, which also reflects the overall/total impact of an article in the research community at large, based on the underlying citation network (diachronically).
BIP!Citations provided by BIP!
popularity
This indicator reflects the "current" impact/attention (the "hype") of an article in the research community at large, based on the underlying citation network.
BIP!Popularity provided by BIP!
influence
This indicator reflects the overall/total impact of an article in the research community at large, based on the underlying citation network (diachronically).
BIP!Influence provided by BIP!
impulse
This indicator reflects the initial momentum of an article directly after its publication, based on the underlying citation network.
BIP!Impulse provided by BIP!
1
Average
Average
Average
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