Synthesis of Novel Aliphatic N-sulfonylamidino Thymine Derivatives by Cu(I)-catalyzed Three-component Coupling Reaction

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Krstulović, Luka; Ismaili, Hamit; Bajić, Miroslav; Višnjevac, Aleksandar; Glavaš-Obrovac, Ljubica; Žinić, Biserka;
(2012)

A series of new aliphatic N-sulfonylamidino thymine derivatives containing nucleobase, N-sulfonyl and amidine pharmacophores in the structure were synthesized by Cu(I)-catalyzed threecomponent coupling of 1-propargyl thymine, benzenesulfonyl azides and amines or a... View more
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