Selective and Specific Inhibition of the Plasmodium falciparum Lysyl-tRNA Synthetase by the Fungal Secondary Metabolite Cladosporin
Hoepfner, Dominic; McNamara, Case W.; Lim, Chek Shik; Studer, Christian; Riedl, Ralph; Aust, Thomas; McCormack, Susan L.; Plouffe, David M.; Meister, Stephan; Schuierer, Sven; Plikat, Uwe; Hartmann, Nicole; Staedtler, Frank; Cotesta, Simona; Schmitt, Esther K.; Petersen, Frank; Supek, Frantisek; Glynne, Richard J.; Tallarico, John A.; Porter, Jeffrey A.; Fishman, Mark C.; Bodenreider, Christophe; Diagana, Thierry T.; Movva, N. Rao; Winzeler, Elizabeth A.;
- Publisher: Elsevier BV
- Journal: Cell Host & Microbe,volume 11,issue 6,pages654-663 (issn: 1931-3128, eissn: 1934-6069)
Related identifiers: , - Subject: Molecular Biology | Immunology and Microbiology(all) | Article | Cancer Research
Summary With renewed calls for malaria eradication, next-generation antimalarials need be active against drug-resistant parasites and efficacious against both liver- and blood-stage infections. We screened a natural product library to identify inhibitors of Plasmodium f... View more
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Genomics Institute Of The Novartis Research Foundation 90%Novartis Institute For Tropical Diseases 90%Genomics Institute of the Novartis Research Foundation United StatesWebsite url: https://www.gnf.nibr.com/90%Novartis Institutes for Biomedical Research ( NIBR ) United States89%Novartis Pharma AG 90%Novartis Institute for Tropical Diseases 90%Genomics Institute of the Novartis Research Foundation ( GNF ) United StatesWebsite url: http://www.gnf.org/90% - Bioentities (3)
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