Enantioselective α‑Aminophosphonate Functionalization of Indole Ring through an Organocatalyzed Friedel–Crafts Reaction

Dataset UNKNOWN
Maestro, Aitor; Martinez de Marigorta, Edorta; Palacios, Francisco; Vicario, Javier;
(2018)
  • Publisher: Figshare
  • Related identifiers: doi: 10.1021/acs.joc.8b02843.s002, doi: 10.1021/acs.joc.8b02843.s003
  • Subject: Molecular Biology | Biotechnology | indole | Plant Biology | derivative | functionalized | catalyze | acid | Genetics | Organocatalyzed | Friedel | phosphoric | α- | Biophysics | Enantioselective | Chiral | Neuroscience | Microbiology | Physiology | Indole Ring | enantioenriched | Functionalization | Aminophosphonate | Biochemistry | imino
    • FOR: 110309 Infectious Diseases | 60506 Virology | 39999 Chemical Sciences not elsewhere classified
    mesheuropmc: heterocyclic compounds

Chiral phosphoric acids efficiently catalyze the asymmetric Friedel–Crafts reaction of several indoles with α-imino­phosphonates to afford enantioenriched hybrid α-amino­phosphonate functionalized indole derivatives.
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